EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.1.1.148 | 0.000028 |
- |
2-(furan-2-yl)-3-hydroxynaphthalene-1,4-dione |
pH 8.0, 37°C |
757894 |
2.1.1.148 | 0.000057 |
- |
ethyl (4R)-2-phenyl-3-([(1-(3-2,2,2-trifluoroacetamido)propyl)-1H-1,2,3-triazol-4-yl]carbonyl)-1,3-thiazolidine-4-carboxylate |
- |
691285 |
2.1.1.148 | 0.0001 |
- |
5-fluoro-2'-deoxyuridine 5'-monophosphate |
inhibited both ThyA and ThyX |
694812 |
2.1.1.148 | 0.00013 |
- |
(heptanoyl[[(4R)-2-phenyl-3-(phenylcarbonyl)-1,3-thiazolidin-4-yl]methyl] amino)acetic acid |
- |
691285 |
2.1.1.148 | 0.000258 |
- |
2-hydroxy-3-propylnaphthalene-1,4-dione |
pH 8.0, 37°C |
757894 |
2.1.1.148 | 0.000367 |
- |
2-hydroxy-3-(4-methoxyphenyl)naphthalene-1,4-dione |
pH 8.0, 37°C |
757894 |
2.1.1.148 | 0.001 |
- |
2-[4-fluoro-3-(trifluoromethyl)phenyl]-3-hydroxynaphthalene-1,4-dione |
pH 8.0, 37°C |
757894 |
2.1.1.148 | 0.001 |
- |
ethyl (4R)-2-phenyl-3-[[1-(2-thiophen-3-ylethyl)-1H-1,2,3-triazol-4-yl]carbonyl]-1,3-thiazolidine-4-carboxylate |
- |
691285 |
2.1.1.148 | 0.002 |
- |
ethyl (4R)-3-([1-[2-(4-fluorophenyl)ethyl]-1H-1,2,3-triazol-4-yl]carbonyl)-2-phenyl-1,3-thiazolidine-4-carboxylate |
- |
691285 |
2.1.1.148 | 0.0035 |
- |
ethyl (4R)-3-[[1-(7-hydroxyheptyl)-1H-1,2,3-triazol-4-yl]carbonyl]-2-phenyl-1,3-thiazolidine-4-carboxylate |
- |
691285 |