EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.17.1.9 | 0.000007 |
- |
azide |
- |
687304 |
1.17.1.9 | 0.0000239 |
- |
azide |
substrate formate, pH 6.5, 30°C |
673381 |
1.17.1.9 | 0.00015 |
- |
azide |
pH 7.0, 37°C, wild-type enzyme |
288102 |
1.17.1.9 | 0.00095 |
- |
azide |
substrate NAD+, pH 6.5, 30°C |
673381 |
1.17.1.9 | 0.0228 |
- |
ADP-beta-D-ribose |
substrate formate, pH 6.5, 30°C |
673381 |
1.17.1.9 | 0.024 |
- |
azide |
pH 7.0, 37°C, mutant enzyme R284Q |
288102 |
1.17.1.9 | 0.0369 |
- |
ADP-beta-D-ribose |
substrate NAD+, pH 6.5, 30°C |
673381 |
1.17.1.9 | 0.053 |
- |
bicarbonate |
substrate formate, pH 6.5, 30°C |
673381 |
1.17.1.9 | 0.06 |
- |
NADH |
substrate NAD+, pH 6.5, 30°C |
673381 |
1.17.1.9 | 0.1175 |
- |
NADH |
at pH 7.5, 25°C |
711549 |