EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.2.3.1 | 0.0000029 |
- |
raloxifene |
- |
691701 |
1.2.3.1 | 0.00009 |
- |
raloxifene |
pH 7.4, 37°C |
741471 |
1.2.3.1 | 0.0004 |
- |
menadione |
substrate vanillin, pH 7.0, 37°C |
699237 |
1.2.3.1 | 0.0004 |
- |
myricetin |
substrate vanillin, pH 7.0, 37°C |
699237 |
1.2.3.1 | 0.0004 |
- |
myricetin |
substrate xanthine, pH 7.0, 37°C |
699237 |
1.2.3.1 | 0.0004 |
- |
quercetin |
substrate vanillin, pH 7.0, 37°C |
699237 |
1.2.3.1 | 0.00062 |
- |
estradiol |
pH 7.4, 37°C |
741471 |
1.2.3.1 | 0.0007 |
- |
quercetin |
substrate phenanthridine, pH 7.0, 37°C |
699237 |
1.2.3.1 | 0.0007 |
- |
quercetin |
substrate xanthine, pH 7.0, 37°C |
699237 |
1.2.3.1 | 0.00094 |
- |
quetiapine |
pH 7.4, 37°C |
741471 |