EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   1.1.1.62 | -999 |
- |
(2,4-dihydroxyphenyl)-phenylmethanone |
value higher than 0.02, pH 7.4, 37°C |
711161 |
| 1.1.1.62 | -999 |
- |
(2,4-dihydroxyphenyl)-phenylmethanone |
value higher than 0.065, pH 7.4, 37°C |
711161 |
| 1.1.1.62 | 0.00000362 |
- |
2-[2-ethyl-3-hydroxy-17-oxoestra-1(10),2,4-trien-16-yl]-N-(pyridin-2-ylmethyl)acetamide |
- |
686263 |
| 1.1.1.62 | 0.000005 |
- |
3-benzyl-2-(2-bromo-3,4,5-trimethoxyphenyl)-8-hydroxy[1]benzothieno[2,3-d]pyrimidin-4(3H)-one |
87% inhibition at 100 nM, 95% inhibition at 0.001 mM. IC50: 5 nM |
670254, 670260 |
| 1.1.1.62 | 0.000005 |
- |
3-benzyl-8-hydroxy-2-(3,4,5-trimethoxyphenyl)[1]benzothieno[2,3-d]pyrimidin-4(3H)-one |
- |
686263 |
| 1.1.1.62 | 0.000005 |
- |
3-benzyl-8-hydroxy-2-(3,4,5-trimethoxyphenyl)[1]benzothieno[2,3-d]pyrimidin-4(3H)-one |
94% inhibition at 100 nM, 99% inhibition at 0.001 mM. IC50: 5 nM |
670254, 670260 |
| 1.1.1.62 | 0.00001 |
- |
(4R,5R)-4-(2-fluorophenyl)-5-[hydroxy(5-phenylthiophen-2-yl)methyl]-1-methylpyrrolidin-2-one |
pH 7.4, 37°C |
740843 |
| 1.1.1.62 | 0.000015 |
- |
(4aS,4bR,10bS,12aS)-8-hydroxy-12a-methyl-9-(2-phenylethyl)-3,4,4a,4b,5,6,10b,11,12,12a-decahydrochrysen-1(2H)-one |
- |
686263 |
| 1.1.1.62 | 0.000016 |
- |
(13S,17R)-3-hydroxy-5',13-dimethyl-4',5',6,7,8,9,11,12,13,14,15,16-dodecahydrospiro[cyclopenta[a]phenanthrene-17,2'-pyran]-6'(3'H)-one |
- |
686533 |
| 1.1.1.62 | 0.000019 |
- |
(13S,17R)-3-hydroxy-4',13-dimethyl-4',5',6,7,8,9,11,12,13,14,15,16-dodecahydrospiro[cyclopenta[a]phenanthrene-17,2'-pyran]-6'(3'H)-one |
- |
686533 |
