EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.3.2.5 | -999 |
- |
more |
inhibition kinetics |
759510 |
2.3.2.5 | 0.000006 |
- |
N-(3,4-dimethoxyphenyl)-N'-[3-(1H-imidazol-1-yl)propyl]thiourea |
pH and temperature not specified in the publication |
759074 |
2.3.2.5 | 0.00002 |
- |
SEN177 |
pH 8.0, 25°C, with enzyme mutant Y115E/Y117E |
759510 |
2.3.2.5 | 0.000023 |
- |
5-(5-[[(3,4-dimethoxyphenyl)sulfanyl]methyl]-1,3,4-oxadiazol-2-yl)-1H-benzimidazole |
pH and temperature not specified in the publication |
759074 |
2.3.2.5 | 0.00006 |
- |
1-(3,4-dimethoxyphenyl)-3-[3-(1H-imidazol-1-yl)propyl]thiourea |
pH 8.0, 30°C |
675310 |
2.3.2.5 | 0.000095 |
- |
PBD150 |
secretory glutaminyl cyclase, at 25°C in 50 mM Tris-HCl, pH 8.0 |
719915 |
2.3.2.5 | 0.000097 |
- |
P150/03 |
pH 8, isoDromeQC |
685085 |
2.3.2.5 | 0.0001 |
- |
PBD150 |
pH 8.0, 30°C |
688518 |
2.3.2.5 | 0.0001 |
- |
PBD150 |
wild type enzyme, in 50 mM Tris, pH 8.0, at 30°C |
719267 |
2.3.2.5 | 0.000101 |
- |
1-Methylimidazole |
pH 7, isoDromeQC |
685085 |