Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2,2'-dipyridyl | IC50 0.029 mM | Homo sapiens | |
4,6-diphenyl-1-hydroxy-pyridine-2-one | IC50 0.0007 mM | Homo sapiens | |
ciclopirox | IC50 0.0006 mM | Homo sapiens | |
Co(C2H3O2)2 | above 0.01 mM | Homo sapiens | |
CuCl2 | above 0.01 mM | Homo sapiens | |
EDTA | IC50 0.0003 mM | Homo sapiens | |
metipirox | IC50 0.0028 mM | Homo sapiens | |
mimosine | IC50 0.0033 mM | Homo sapiens | |
Mn(C2H3O2)2 | above 0.001 mM | Homo sapiens | |
additional information | partial reconstitution of chelator inhibited activity with CuCl2 or Zn(C2H3O2)2 | Homo sapiens | |
Ni(C2H3O2)2 | above 0.001 mM | Homo sapiens | |
Zn(C2H3O2)2 | above 0.01 mM | Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Fe2+ | 1.5-fold activation at 0.001 mM | Homo sapiens | |
Fe3+ | 1.5-fold activation at 0.001 mM | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
HeLa-S3 cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
N'-(4-aminobutyl)lysine + electron donor + O2 | i.e. deoxyhypusine | Homo sapiens | N'-(4-amino-2-hydroxybutyl)lysine + oxidized electron donor + H2O | i.e. hypusine | ? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.5 | - |
assay in 50 mM sodium phosphate buffer | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0003 | - |
IC50 0.0003 mM | Homo sapiens | EDTA | |
0.0006 | - |
IC50 0.0006 mM | Homo sapiens | ciclopirox | |
0.0007 | - |
IC50 0.0007 mM | Homo sapiens | 4,6-diphenyl-1-hydroxy-pyridine-2-one | |
0.0028 | - |
IC50 0.0028 mM | Homo sapiens | metipirox | |
0.0033 | - |
IC50 0.0033 mM | Homo sapiens | mimosine | |
0.029 | - |
IC50 0.029 mM | Homo sapiens | 2,2'-dipyridyl |